BAR 501 impurity

CAS No. 1632118-70-7

BAR 501 impurity( —— )

Catalog No. M22739 CAS No. 1632118-70-7

BAR501 impurity is an impurity found in the preparation of BAR501 that acts as an agonist of the G protein-coupled bile acid-activated receptor (GP-BAR1).?

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    BAR 501 impurity
  • Note
    Research use only, not for human use.
  • Brief Description
    BAR501 impurity is an impurity found in the preparation of BAR501 that acts as an agonist of the G protein-coupled bile acid-activated receptor (GP-BAR1).?
  • Description
    BAR501 impurity is an impurity found in the preparation of BAR501 that acts as an agonist of the G protein-coupled bile acid-activated receptor (GP-BAR1).?BAR501 impurity (10 μM) induces a 150% increase in luciferase activity in a GP-BAR1 reporter gene assay.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    GPCR19
  • Recptor
    GPBAR1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1632118-70-7
  • Formula Weight
    406.6
  • Molecular Formula
    C26H46O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    [H][C@@]12CC[C@H]([C@H](C)CCCO)[C@@]1(C)CC[C@@]1([H])[C@@]2([H])[C@H](O)[C@@H](CC)[C@]2([H])C[C@H](O)CC[C@]12C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Renga B, et al. Reversal of Endothelial Dysfunction by GPBAR1 Agonism in Portal Hypertension Involves a AKT/FOXOA1 Dependent Regulation of H2S Generation and Endothelin-1.
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